Difference in mGluR5 interaction between positive allosteric modulators from two structural classes.

David L Williams; Julie A O'Brien; Wei Lemaire; Tsing-Bau Chen; Raymond S L Chang; Marlene A Jacobson; Sookhee N Ha; David D Wisnoski; Craig W Lindsley; Cyrille Sur; Mark E Duggan; Douglas J Pettibone; P Jeffrey Conn

doi:10.1196/annals.1300.059

PubMed · 14684495

Difference in mGluR5 interaction between positive allosteric modulators from two structural classes.

David L Williams·Julie A O'Brien·Wei Lemaire·Tsing-Bau Chen·Raymond S L Chang·Marlene A Jacobson·Sookhee N Ha·David D Wisnoski·Craig W Lindsley·Cyrille Sur·Mark E Duggan·Douglas J Pettibone·P Jeffrey Conn

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Animals Benzamides Binding Sites CHO Cells Cricetinae Excitatory Amino Acid Agonists Excitatory Amino Acid Antagonists Glycine Humans Hydrazines Phthalimides Rats Receptor, Metabotropic Glutamate 5 Receptors, Metabotropic Glutamate Resorcinols Structure-Activity Relationship Journal Article

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David L Williams, Julie A O'Brien, Wei Lemaire, Tsing-Bau Chen, Raymond S L Chang, Marlene A Jacobson, Sookhee N Ha, David D Wisnoski, Craig W Lindsley, Cyrille Sur, Mark E Duggan, Douglas J Pettibone, P Jeffrey Conn. 2003. Difference in mGluR5 interaction between positive allosteric modulators from two structural classes.. https://doi.org/10.1196/annals.1300.059

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