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PubMed · 12498013

Eletriptan Pfizer.

Paul J L M Strijbos·Andrew A Parsons·Anders Fugelli
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Abstract

Pfizer has developed and launched eletriptan, a 5-HT1B/1D agonist, for the potential treatment of migraine with and without aura. Eletriptan has 6-fold greater affinity for the 5-HT1D receptor than sumatriptan, and a 3-fold greater affinity for the 5-HT1B receptor [249570]. Eletriptan pharmacology has also been evaluated in vitro in comparison with zolmitriptan (AstraZeneca plc) and naratriptan (GlaxoSmithKline plc) [290116].

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Paul J L M Strijbos, Andrew A Parsons, Anders Fugelli. 2002. Eletriptan Pfizer.. https://pubmed.ncbi.nlm.nih.gov/12498013/

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