Dissolution rate limited absorption in man. Factors influencing drug absorption from prolonged-release dosage form.
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Biomedical subjects
Publications and source records attributed to G Levy.
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The free fraction of d-propoxyphene in the plasma of normal subjects is 0.24 +/- 0.02 (mean +/- S.D.) and is not concentration dependent in the usual therapeutic and toxic conentration range. Renal failure and relatively high concentrations of d-norpropoxyphene, the major metabolite of d-propoxyphene, have no significant effect on the plasma protein binding of d-propoxyphene.
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