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PubMed · 16375751

A2B adenosine receptor antagonists: recent developments.

Barbara Cacciari·Giorgia Pastorin·Chiara Bolcato·Giampiero Spalluto·Magdalena Bacilieri·Stefano Moro
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Abstract

There are pharmacological evidences that A(2B) receptors are involved in inflammatory processes, such as asthma. For this reason, many efforts has been made for identifying selective A(2B) antagonists as anti-asthmatic agents. The updated material related to this field has been rationalised and arranged in order to offer an overview of the topic.

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Adenosine A2 Receptor AntagonistsAmino Acid SequenceAnimalsAnti-Asthmatic AgentsAnti-Inflammatory AgentsAsthmaBinding SitesDrug DesignHumansMolecular Sequence DataQuinazolinesTriazolesXanthinesJournal ArticleReview

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Barbara Cacciari, Giorgia Pastorin, Chiara Bolcato, Giampiero Spalluto, Magdalena Bacilieri, Stefano Moro. 2005. A2B adenosine receptor antagonists: recent developments.. https://doi.org/10.2174/138955705774933374

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Adenosine A2 Receptor Antagonists↗
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